What are benzodiazepines, and how do they work (mechanism of action)? Benzodiazepines are man-made medications that cause mild to severe depression of the nerves within the brain (central nervous system) and sedation (drowsiness). Seizures, anxiety, and other diseases that require benzodiazepine treatment may be caused by excessive activity of nerves in the brain. These drugs …
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What is Intermezzo? What is zolpidem used for? Intermezzo contains a low dose of zolpidem, the same active ingredient in Ambien. Zolpidem belongs to a class of drugs called sedatives or hypnotics. Zolpidem shares some characteristics of a family of sedatives called benzodiazepines which includes diazepam (Valium). Benzodiazepines cause sedation, muscle relaxation, act as anticonvulsants (antiseizure medications), and reduce anxiety. …
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What is zaleplon, and how does it work (mechanism of action)? Zaleplon is a hypnotic (a medication that induces sleep) that is used for treating insomnia. It is chemically unrelated to the benzodiazepine class of medications for sleep, for example, lorazepam (Ativan), oxazepam (Serax), flurazepam (Dalmane), triazolam (Halcion), and temazepam (Restoril), but it has similar effects because it attaches to …
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What are oral caffeine tablets, and how do they work (mechanism of action)? Caffeine acts as a stimulant of the nervous system by inhibiting the enzyme phosphodiesterase, just like theophylline and aminophylline. Inhibiting this enzyme leads to increased formation of the proteins which causes release of stimulating chemical signals known as neurotransmitters. These neurotransmitters bind to various sites in the …
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What is armodafinil, and how does it work (mechanism of action)? Armodafinil is an oral drug that is used to promote wakefulness. It is similar to modafinil (Provigil). Like amphetamines, armodafinil promotes wakefulness by stimuatIng the brain; however, the exact mechanism of action of armodafinil is unknown. Armodafinil may work by increasing the amount of dopamine (a chemical neurotransmitter that …
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Klonopin vs. temazepam: What’s the difference? Klonopin (clonazepam) and Restoril (temazepam) are benzodiazepines used to treat anxiety. Klonopin is primarily used for treating panic disorder and preventing certain types of seizures such as those caused by Lennox-Gastaut syndrome. Temazepam is used to treat symptoms of insomnia. A brand name for clonazepam is Klonopin. A brand name for temazepam is Restoril. …
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Clonazepam vs. Ambien: What’s the difference? Clonazepam and Ambien (zolpidem) are used to treat insomnia. Clonazepam is primarily used for treating panic disorder and preventing certain types of seizures, treating Lennox-Gastaut syndrome, and providing short-term relief of anxiety symptoms. A brand name for clonazepam is Klonopin. Clonazepam and Ambien belong to different drug classes. Clonazepam is a benzodiazepine, which include …
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What is Rozerem, and how does it work (mechanism of action)? Ramelteon is an oral drug that promotes falling asleep and is used for treating insomnia. It acts by stimulating receptors for melatonin in the brain. Melatonin and its receptors control the circadian rhythm of the body which controls the sleep/wake cycle. Unlike many drugs used for treating insomnia, ramelteon …
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What is triazolam, and how does it work (mechanism of action)? Triazolam is a drug that is used to promote sleep in individuals who have difficulty sleeping (insomnia). It is in the benzodiazepine family of drugs, the same family that includes diazepam (Valium), alprazolam (Xanax), clonazepam (Klonopin), flurazepam (Dalmane), lorazepam (Ativan), and others. Insomnia is believed often to be the …
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What is melatonin, and how does it work (mechanism of action)? Melatonin is a natural hormone produced by the pineal gland in the body. Commercially available melatonin that is sold as medicine is produced in the laboratory. Melatonin regulates sleep-wake cycle. Check with your healthcare professional before using herbs or other supplements. What brand names are available for melatonin? N/A …
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